Bortezomib

Generic Name: bortezomib

Proteasome Inhibitor [EPC]Over-the-Counter (OTC)

Brand Names:

Bortezomib

Bortezomib is a proteasome inhibitor indicated for treatment of adult patients with multiple myeloma and mantle cell lymphoma.

Overview

Bortezomib is a proteasome inhibitor indicated for treatment of adult patients with multiple myeloma and mantle cell lymphoma.

Uses

Indicated for treatment of adult patients with multiple myeloma and mantle cell lymphoma.

Dosage

The recommended starting dose is 1.3 mg/m2 administered as a 3 to 5 second bolus intravenous injection or subcutaneous injection. For intravenous or subcutaneous use only.

Side Effects

Most commonly reported adverse reactions (20% or more) include nausea, diarrhea, thrombocytopenia, neutropenia, peripheral neuropathy, fatigue, neuralgia, anemia, leukopenia, constipation, vomiting, lymphopenia, rash, pyrexia, and anorexia.

Warnings

Peripheral neuropathy, hypotension, cardiac toxicity, pulmonary toxicity, posterior reversible encephalopathy syndrome, gastrointestinal toxicity, thrombocytopenia/neutropenia, tumor lysis syndrome, hepatic toxicity, thrombotic microangiopathy, and embryo-fetal toxicity require monitoring and potential dose modification. Contraindicated in patients with hypersensitivity to bortezomib, boron, or mannitol, and for intrathecal administration.

Storage

Store unopened vials in original package protected from light. Administer reconstituted product within eight hours.

Frequently Asked Questions

What is Bortezomib used for?

Indicated for treatment of adult patients with multiple myeloma and mantle cell lymphoma.

What are the side effects of Bortezomib?

Most commonly reported adverse reactions (20% or more) include nausea, diarrhea, thrombocytopenia, neutropenia, peripheral neuropathy, fatigue, neuralgia, anemia, leukopenia, constipation, vomiting, lymphopenia, rash, pyrexia, and anorexia.

What are the important warnings for Bortezomib?

Peripheral neuropathy, hypotension, cardiac toxicity, pulmonary toxicity, posterior reversible encephalopathy syndrome, gastrointestinal toxicity, thrombocytopenia/neutropenia, tumor lysis syndrome, hepatic toxicity, thrombotic microangiopathy, and embryo-fetal toxicity require monitoring and potential dose modification. Contraindicated in patients with hypersensitivity to bortezomib, boron, or mannitol, and for intrathecal administration.

Related Medications

Medical Disclaimer

This drug information is for educational purposes only and should not replace professional medical advice. Drug information is sourced from the FDA National Drug Code Directory and Structured Product Labeling. Always consult with a healthcare provider before starting, stopping, or changing any medication.