Norgestrel And Ethinyl Estradiol

Generic Name: norgestrel and ethinyl estradiol

Over-the-Counter (OTC)

Brand Names:

Cryselle

Norgestrel and ethinyl estradiol is a combination oral contraceptive containing 0.3 mg norgestrel and 0.03 mg ethinyl estradiol per active tablet, indicated for pregnancy prevention.

Overview

Norgestrel and ethinyl estradiol is a combination oral contraceptive containing 0.3 mg norgestrel and 0.03 mg ethinyl estradiol per active tablet, indicated for pregnancy prevention.

Uses

Indicated for use by females of reproductive potential to prevent pregnancy, with approximately 1 pregnancy per 100 women-years of use.

Dosage

One white active tablet daily for 21 consecutive days, followed by one light green inert tablet daily for 7 consecutive days.

Side Effects

Common reactions include weight changes (11% increase), cervical erosion (9%), acne (4%), dysmenorrhea (4%), and vaginal discharge (4%).

Interactions

Multiple interactions documented including enzyme inducers, bile acid sequestrants, CYP3A4 inhibitors, and effects on other drug metabolism.

Warnings

Cigarette smoking increases the risk of serious cardiovascular events from combination oral contraceptive use. Contraindicated in smokers over 35, those with history of blood clots, cerebrovascular/coronary disease, uncontrolled hypertension, liver tumors, breast cancer, and those taking specific Hepatitis C medications.

Pregnancy

Not indicated during pregnancy. Discontinue if pregnancy is confirmed. Inadvertent early exposure shows no increased birth defect risk. Nursing mothers advised to use alternative contraception; COCs may reduce milk production.

Storage

Store at 68-77 degrees F (20-25 degrees C). Keep away from light and out of children's reach.

Frequently Asked Questions

What is Norgestrel And Ethinyl Estradiol used for?

Indicated for use by females of reproductive potential to prevent pregnancy, with approximately 1 pregnancy per 100 women-years of use.

What are the side effects of Norgestrel And Ethinyl Estradiol?

Common reactions include weight changes (11% increase), cervical erosion (9%), acne (4%), dysmenorrhea (4%), and vaginal discharge (4%).

Can I take Norgestrel And Ethinyl Estradiol during pregnancy?

Not indicated during pregnancy. Discontinue if pregnancy is confirmed. Inadvertent early exposure shows no increased birth defect risk. Nursing mothers advised to use alternative contraception; COCs may reduce milk production.

What are the important warnings for Norgestrel And Ethinyl Estradiol?

Cigarette smoking increases the risk of serious cardiovascular events from combination oral contraceptive use. Contraindicated in smokers over 35, those with history of blood clots, cerebrovascular/coronary disease, uncontrolled hypertension, liver tumors, breast cancer, and those taking specific Hepatitis C medications.

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Medical Disclaimer

This drug information is for educational purposes only and should not replace professional medical advice. Drug information is sourced from the FDA National Drug Code Directory and Structured Product Labeling. Always consult with a healthcare provider before starting, stopping, or changing any medication.